Klomipramin je [[inhibitor preuzimanja|blokator]] sledećih [[membranski transportni protein|transportera]]:<ref name="pmid11454918">{{cite journal | author author1=Millan MJ, |author2=Gobert A, |author3=Lejeune F, |author4=''et al.'' | title = S33005, a novel ligand at both serotonin and norepinephrine transporters: I. Receptor binding, electrophysiological, and neurochemical profile in comparison with venlafaxine, reboxetine, citalopram, and clomipramine | journal = The Journal of Pharmacology and Experimental Therapeutics | volume = 298 | issue = 2 | pages = 565–80 | year = 2001 | month = August | pmid = 11454918 | doi = | url = http://jpet.aspetjournals.org/cgi/pmidlookup?view=long&pmid=11454918}}</ref>
On je [[antagonist (farmakologija)|antagonist]]/[[inverzni agonist]] sledećih [[receptor (biohemija)|receptora]]:<ref name="pmid11454918"/><ref name="pmid7680751">{{cite journal | author vauthors=Monsma FJ, Shen Y, Ward RP, Hamblin MW, Sibley DR | title = Cloning and expression of a novel serotonin receptor with high affinity for tricyclic psychotropic drugs | journal = Molecular Pharmacology | volume = 43 | issue = 3 | pages = 320–7 | year = 1993 | month = March | pmid = 7680751 | doi = | url = http://molpharm.aspetjournals.org/cgi/pmidlookup?view=long&pmid=7680751}}</ref><ref name="pmid8397408">{{cite journal | author author1=Ruat M, |author2=Traiffort E, |author3=Leurs R, |author4=''et al.'' | title = Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation | journal = Proceedings of the National Academy of Sciences of the United States of America | volume = 90 | issue = 18 | pages = 8547–51 | year = 1993 | month = September | pmid = 8397408 | pmc = 47394 | doi = 10.1073/pnas.90.18.8547| url = }}</ref><ref name="pmid9686407">{{cite journal | author author1=Toll L, |author2=Berzetei-Gurske IP, |author3=Polgar WE, |author4=''et al.'' | title = Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications | journal = NIDA Research Monograph | volume = 178 | issue = | pages = 440–66 | year = 1998 | month = March | pmid = 9686407 | doi = | url = }}</ref>
