Ro10-5824
Ro10-5824 je lek koji deluje kao dopaminski agonist. On je selektivni parcijalni agonist D4 podtipa. Ro10-5824 deluje kao kognitivni pojačivač u životinjskim studijama.[1][2]
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IUPAC ime | |
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2-metil-5-[(4-fenil-3,6-dihidro-2H-piridin-1-il)metil]pirimidin-4-amin | |
Identifikatori | |
CAS broj | 189744-46-5 ![]() |
ATC kod | none |
PubChem | CID 16759175 |
Hemijski podaci | |
Formula | C17H20N4 |
Molarna masa | 280,367 g/mol |
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Reference
уреди- ^ Powell SB, Paulus MP, Hartman DS, Godel T, Geyer MA (2003). „RO-10-5824 is a selective dopamine D4 receptor agonist that increases novel object exploration in C57 mice”. Neuropharmacology. 44 (4): 473—81. PMID 12646284. doi:10.1016/S0028-3908(02)00412-4.
- ^ Newman-Tancredi A, Heusler P, Martel JC, Ormière AM, Leduc N, Cussac D (2008). „Agonist and antagonist properties of antipsychotics at human dopamine D4.4 receptors: G-protein activation and K+ channel modulation in transfected cells”. The International Journal of Neuropsychopharmacology / Official Scientific Journal of the Collegium Internationale Neuropsychopharmacologicum (CINP). 11 (3): 293—307. PMID 17897483. doi:10.1017/S1461145707008061.